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The Phosphinoboration of N-Heterocycles.

Author
Abstract
:

The addition of phosphinoboronate ester Ph PBpin (pin=1,2-O C Me ) (1) to a number of different N-heterocycles has been investigated. Reaction of 1 with pyridine resulted in highly selective formation of the corresponding 1,4-addition product, with addition of the electron-deficient Bpin group to the pyridine nitrogen atom and the phosphido group to the para carbon atom. Conversely, reactions of para-substituted pyridine derivatives occurred predominately to afford 1,2-addition products while quinoline reacted to afford the 1,2-adduct which ultimately isomerized to afford the corresponding 1,4-addition product. Preliminary computational studies have been undertaken to explore possible pathways for these transformations including transfer of the PPh anion from [B(PPh ) pin] to the 4-position of a borenium/boronium activated pyridine and concerted pathways for 1,2-addition via intramolecular nucleophilic attack of PPh at C2 of a Ph PBpin-coordinated pyridine via a four-centered transition state and intramolecular transfer of PPh to the 2-position of a boron-activated pyridine in a phosphido-bridged dimer involving a six-centered transition state.

Year of Publication
:
2017
Journal
:
Chemistry (Weinheim an der Bergstrasse, Germany)
Volume
:
23
Issue
:
58
Number of Pages
:
14485-14499
Date Published
:
2017
ISSN Number
:
0947-6539
DOI
:
10.1002/chem.201702203
Short Title
:
Chemistry
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